SCHEMBL22628754

SCHEMBL22628754

C=CC(=O)OCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)CCOc1ccc2cc(-c3cccnc3)oc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.38
APP P05067 1/20 0.36
THRB P10828 1/20 0.34
NAMPT P43490 1/20 0.34
CYP19A1 P11511 3/20 0.34
MAPT P10636 3/20 0.34
KDM4E B2RXH2 5/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
PPARG P37231 2/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
PPARA Q07869 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
PRKDC P78527 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21735738 0.90 SIGMAR1 (0.37) SIGMAR1APPTHRBNAMPTCYP19A1
SCHEMBL21735560 0.89 THRB (0.43) SIGMAR1THRBMAPTKDM4EALDH1A1
SCHEMBL21734956 0.89 SIGMAR1 (0.40) SIGMAR1APPTHRBNAMPTCYP19A1
SCHEMBL21735359 0.88 SIGMAR1 (0.38) SIGMAR1APPNAMPTCYP19A1MAPT
SCHEMBL22628923 0.87 CYP2E1 (0.32) CYP19A1MAPTKDM4EKMT2AMEN1
SCHEMBL21735100 0.86 APP (0.37) SIGMAR1APPCYP19A1MAPTKDM4E
SCHEMBL21735790 0.83 HDAC1 (0.37) THRBNAMPTCYP19A1MAPTKDM4E
SCHEMBL21735390 0.82 THRB (0.39) SIGMAR1THRBMAPTKDM4EALDH1A1
SCHEMBL21735223 0.82 CYP19A1 (0.36) SIGMAR1APPCYP19A1MAPTKDM4E
SCHEMBL22625065 0.81 NPC1 (0.54) MAPTKDM4EKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3583091-B1 HYDROPHOBIC COMPOUNDS FOR OPTICALLY ACTIVE DEVICES MERCK PATENT GMBH (DE) 2020-11-04 EP disclosed