SCHEMBL22643116

SCHEMBL22643116

Cc1ccc(-c2cnn(C(=O)CC(C)C)c2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.47
CTSK P43235 1/20 0.47
KCNH2 Q12809 5/20 0.45
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
GRIN2B Q13224 7/20 0.40
NAMPT P43490 1/20 0.38
KMO O15229 2/20 0.37
LMNA P02545 1/20 0.36
MET P08581 1/20 0.35
NPY2R P49146 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19368384 0.86 CTSC (0.53) CTSCCTSKKCNH2GRIN2BNAMPT
SCHEMBL22643394 0.82 CTSC (0.47) CTSCKCNH2AKR1C3AKR1C2GRIN2B
SCHEMBL22642946 0.81 KCNH2 (0.47) CTSCCTSKKCNH2AKR1C3AKR1C2
SCHEMBL22643135 0.75 KCNH2 (0.58) KCNH2GRIN2B
SCHEMBL22643282 0.72 CTSK (0.49) CTSCCTSKKCNH2GRIN2B
SCHEMBL13036109 0.70 KCNH2 (0.59) KCNH2AURKB
SCHEMBL22642936 0.70 KCNH2 (0.53) CTSCCTSKKCNH2GRIN2BNAMPT
SCHEMBL19998601 0.70 KCNH2 (0.62) KCNH2GRIN2B
SCHEMBL19368289 0.69 CTSC (0.52) CTSCCTSKKCNH2GRIN2B
SCHEMBL19155286 0.69 CTSK (0.48) CTSCCTSKKCNH2GRIN2BNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970283-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-11-11 EP disclosed