SCHEMBL22644241

SCHEMBL22644241

CC(C)COc1ccc([C@]23CC4CC(C[C@H](C4)C2)C3)c(F)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.36
RARA P10276 2/20 0.36
RARB P10826 2/20 0.36
RARG P13631 2/20 0.36
GAA P10253 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HTR2C P28335 1/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
HTT P42858 1/20 0.33
RAD52 P43351 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
LMNA P02545 2/20 0.32
VDR P11473 1/20 0.32
IGF1R P08069 1/20 0.32
NR1I2 O75469 1/20 0.32
PGR P06401 1/20 0.32
HSPD1 P10809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22644229 0.85 RARA (0.39) RARARARBRARGGAAMEN1
SCHEMBL24559482 0.84 RARB (0.41) RARARARBRARGGAAMEN1
SCHEMBL15046513 0.79 RARA (0.43) RARARARBRARGALDH1A1MEN1
SCHEMBL24559663 0.76 RARB (0.36) RARARARBRARGGAAALDH1A1
SCHEMBL22635921 0.76 RARA (0.35) RARARARBRARGGAAALDH1A1
SCHEMBL24559474 0.76 RARA (0.35) RARARARBRARGGAAALDH1A1
SCHEMBL22644213 0.76 PPARG (0.33) RARARARBRARGALDH1A1HTR2C
SCHEMBL29240603 0.76 PPARG (0.33) RARARARBRARGALDH1A1HTR2C
SCHEMBL22644230 0.76 RARA (0.35) RARARARBRARGGAAALDH1A1
SCHEMBL24559483 0.76 APP (0.36) RARARARBRARGHTR2CIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020225270-A1 DIAMONDOID COMPOUNDS MERCK PATENT GMBH (DE) 2020-11-12 WO disclosed