SCHEMBL22647948

SCHEMBL22647948

O=C(O)c1ccc(C2CC2)c(SNc2cc(-c3ccns3)c(Cl)cc2-c2ccccn2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 2/20 0.36
DHODH Q02127 2/20 0.34
PRSS12 P56730 1/20 0.34
RORC P51449 4/20 0.33
PFKFB3 Q16875 1/20 0.33
CREBBP Q92793 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KDM6B O15054 1/20 0.33
KDM4A O75164 1/20 0.33
KDM5C P41229 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22647978 0.90 RORC (0.35) NTRK1DHODHPRSS12RORCPFKFB3
SCHEMBL22637297 0.85 PFKFB3 (0.41) NTRK1PFKFB3KDM4EMEN1ALDH1A1
SCHEMBL29430649 0.85 PFKFB3 (0.41) NTRK1PFKFB3KDM4EMEN1ALDH1A1
SCHEMBL22647986 0.84 NTRK1 (0.37) NTRK1DHODHRORCCREBBPKDM4C
SCHEMBL22648195 0.83 NTRK1 (0.36) NTRK1DHODHRORCCREBBP
SCHEMBL22647920 0.83 RORC (0.33) RORCCREBBPKDM4C
SCHEMBL22647935 0.83 NTRK1 (0.37) NTRK1DHODHRORCCREBBPKDM4E
SCHEMBL22647973 0.82 NTRK1 (0.35) NTRK1DHODHRORCCREBBPKDM4E
SCHEMBL22647968 0.81 NTRK1 (0.38) NTRK1DHODHRORCCREBBPKDM4E
SCHEMBL24929582 0.81 KMO (0.33) KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020225569-A1 PHENYL-SULFAMOYL.BENZOYC ACIDS AS ERAP1 MODULATORS Grey Wolf Therapeutics Limited (GB) 2020-11-12 WO disclosed