SCHEMBL22648398

SCHEMBL22648398

CC(C)(C)NC(=O)Nc1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.67
KMT2A Q03164 5/20 0.62
RAB9A P51151 4/20 0.62
MEN1 O00255 4/20 0.62
NPC1 O15118 2/20 0.62
TAAR1 Q96RJ0 2/20 0.58
SMN1; SMN2 Q16637 3/20 0.57
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
TP53 P04637 1/20 0.57
GAA P10253 1/20 0.57
HPGD P15428 1/20 0.57
CASP1 P29466 1/20 0.57
CASP7 P55210 1/20 0.57
HSD17B10 Q99714 1/20 0.57
PKM P14618 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
NAMPT P43490 1/20 0.49
HTT P42858 1/20 0.49
SMARCA2 P51531 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13756247 0.86 RAB9A (0.81) KMT2ARAB9AMEN1NPC1SMN1; SMN2
SCHEMBL10756539 0.83 MDM2 (0.50) MDM2KMT2ARAB9AMEN1NPC1
SCHEMBL10854635 0.83 MDM2 (0.55) MDM2KMT2ARAB9AMEN1NPC1
SCHEMBL10020286 0.81 MDM2 (1.00) MDM2KMT2ARAB9AMEN1TAAR1
SCHEMBL10625584 0.80 NPC1 (0.53) MDM2KMT2ARAB9AMEN1NPC1
SCHEMBL9285165 0.80 NPC1 (0.67) KMT2ARAB9AMEN1NPC1TAAR1
SCHEMBL31668740 0.79 MDM2 (0.95) MDM2KMT2ARAB9AMEN1TAAR1
SCHEMBL12156880 0.79 RAB9A (0.62) KMT2ARAB9AMEN1NPC1TAAR1
SCHEMBL5852111 0.78 RAB9A (0.70) KMT2ARAB9AMEN1NPC1SMN1; SMN2
SCHEMBL15946352 0.78 EPHX2 (0.72) KMT2ARAB9AMEN1NPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION XBP1, RNASE1, ERN1 MDM2 2218/4885KMT2A 3822/4885RAB9A 2652/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.