SCHEMBL22650372

SCHEMBL22650372

CC(C)n1cnc2c(F)nc(-c3nc(Cl)ncc3F)cc21

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.36
CCNA2 P20248 6/20 0.34
CDK2 P24941 6/20 0.34
CDK5 Q00535 6/20 0.34
CDK5R1 Q15078 6/20 0.34
CCNA1 P78396 5/20 0.34
DYRK1A Q13627 5/20 0.34
CDK4 P11802 8/20 0.34
CCND1 P24385 8/20 0.34
CCND3 P30281 7/20 0.34
CDK6 Q00534 7/20 0.34
HTR3A P46098 1/20 0.31
CCNT1 O60563 1/20 0.31
CDK9 P50750 1/20 0.31
GABRA2 P47869 1/20 0.31
MAPK14 Q16539 1/20 0.31
TGFBR1 P36897 1/20 0.31
TGFBR2 P37173 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650364 0.90 CDK4 (0.37) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL22650360 0.89 SMN1; SMN2 (0.41) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL22650721 0.86 SMN1; SMN2 (0.34) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL24632941 0.81 CDK4 (0.43) SMN1; SMN2CCNA2CDK2CDK4CCND1
SCHEMBL29491131 0.79 MAPK14 (0.40) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL22650600 0.79 MAPK14 (0.40) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL22650746 0.76 SMN1; SMN2 (0.45) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL29491171 0.76 SMN1; SMN2 (0.45) SMN1; SMN2CCNA2CDK2CDK5CDK5R1
SCHEMBL30888943 0.76 CDK4 (0.50) CCNA2CDK2CDK4CCND1CCND3
SCHEMBL19209861 0.71 SMN1; SMN2 (0.35) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed