SCHEMBL22650721

SCHEMBL22650721

COc1nc(-c2nc(Cl)ncc2F)cc2c1ncn2C(C)C

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
GAA P10253 1/20 0.33
CCNA2 P20248 2/20 0.31
CDK2 P24941 2/20 0.31
CCNA1 P78396 2/20 0.31
CDK5 Q00535 2/20 0.31
DYRK1A Q13627 2/20 0.31
CDK5R1 Q15078 2/20 0.31
CDK4 P11802 6/20 0.31
CCND1 P24385 6/20 0.31
CCND3 P30281 5/20 0.31
CDK6 Q00534 5/20 0.31
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650372 0.86 SMN1; SMN2 (0.36) SMN1; SMN2CCNA2CDK2CCNA1CDK5
SCHEMBL22650727 0.83 ALDH1A1 (0.33) ALDH1A1HTTGAA
SCHEMBL22650586 0.81 EGFR (0.39) CCNA2CDK2CDK5DYRK1ACDK5R1
SCHEMBL22650407 0.78 L3MBTL1 (0.37) SMN1; SMN2L3MBTL1CCNA2CDK2CCNA1
SCHEMBL24632941 0.78 CDK4 (0.43) SMN1; SMN2CCNA2CDK2CDK4CCND1
SCHEMBL22650364 0.77 CDK4 (0.37) SMN1; SMN2CCNA2CDK2CCNA1CDK5
SCHEMBL22650360 0.76 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1CCNA2CDK2CCNA1
SCHEMBL22650358 0.75 EGFR (0.33) ALDH1A1GAACCNA2CDK2CDK4
SCHEMBL30888943 0.72 CDK4 (0.50) CCNA2CDK2CDK4CCND1CCND3
SCHEMBL27445903 0.70 L3MBTL1 (0.46) SMN1; SMN2L3MBTL1CDK2CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed