SCHEMBL22650552

SCHEMBL22650552

CC(C)n1cnc2c1CN(c1nc(Nc3ccc(N4CCCNC4=O)cc3)ncc1F)CC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.53
CCND1 P24385 4/20 0.53
CDK6 Q00534 2/20 0.53
BMPR2 Q13873 1/20 0.38
JAK2 O60674 9/20 0.37
JAK1 P23458 7/20 0.37
TYK2 P29597 7/20 0.37
JAK3 P52333 7/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RPS6KA6 Q9UK32 2/20 0.37
CDK2 P24941 3/20 0.37
CCNA2 P20248 2/20 0.37
BRD4 O60885 1/20 0.36
KCNH2 Q12809 1/20 0.35
CCND2 P30279 1/20 0.35
CCND3 P30281 1/20 0.35
SYK P43405 1/20 0.34
CDK1 P06493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650556 0.87 CDK4 (0.52) CDK4CCND1CDK6BMPR2JAK2
SCHEMBL22650753 0.85 CDK4 (0.51) CDK4CCND1CDK6BMPR2JAK2
SCHEMBL22650754 0.85 CDK4 (0.51) CDK4CCND1CDK6BMPR2JAK2
SCHEMBL22650761 0.85 CDK4 (0.51) CDK4CCND1CDK6BMPR2JAK2
SCHEMBL22650551 0.79 CDK6 (0.52) CDK4CCND1CDK6JAK2NPC1
SCHEMBL22650445 0.78 CDK4 (0.60) CDK4CCND1CDK6CDK2CCNA2
SCHEMBL22650544 0.78 CDK4 (0.56) CDK4CCND1CDK6BMPR2JAK2
SCHEMBL22650553 0.77 CDK6 (0.51) CDK4CCND1CDK6BMPR2CDK2
SCHEMBL22650444 0.77 CDK4 (0.50) CDK4CCND1CDK6CDK2CCNA2
SCHEMBL22650545 0.77 CDK4 (0.55) CDK4CCND1CDK6BMPR2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed