SCHEMBL22650551

SCHEMBL22650551

CC(C)n1cnc2c1CN(c1nc(Nc3ccc(N4CCCC(N(C)C)C4)cc3)ncc1F)CC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 8/20 0.52
CDK4 P11802 7/20 0.52
CCND1 P24385 2/20 0.52
CDK2 P24941 8/20 0.39
CDK1 P06493 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FGFR4 P22455 1/20 0.38
CDK5 Q00535 4/20 0.36
CSF1R P07333 4/20 0.36
CCNK O75909 3/20 0.36
CCNA2 P20248 3/20 0.36
CDK7 P50613 3/20 0.36
CDK9 P50750 3/20 0.36
CCNH P51946 3/20 0.36
CDK5R1 Q15078 3/20 0.36
JAK2 O60674 2/20 0.36
BRD4 O60885 2/20 0.36
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650761 0.85 CDK4 (0.51) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650753 0.81 CDK4 (0.51) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650754 0.81 CDK4 (0.51) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650552 0.79 CDK4 (0.53) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650556 0.76 CDK4 (0.52) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650762 0.75 CDK6 (0.67) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650544 0.75 CDK4 (0.56) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650545 0.74 CDK4 (0.55) CDK6CDK4CCND1CDK2CDK1
SCHEMBL22650749 0.69 CDK4 (0.54) CDK6CDK4CCND1SMN1; SMN2
SCHEMBL22650447 0.69 CDK4 (0.60) CDK6CDK4CCND1CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed