SCHEMBL22650753

SCHEMBL22650753

CC(C)n1cnc2c1CN(c1nc(Nc3ccc(N4CCCC(N)C4=O)cc3)ncc1F)CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.51
CCND1 P24385 4/20 0.51
CDK6 Q00534 2/20 0.51
BMPR2 Q13873 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CDK2 P24941 4/20 0.35
RPS6KA6 Q9UK32 2/20 0.34
EGFR P00533 1/20 0.34
FYN P06241 1/20 0.34
PDGFRB P09619 1/20 0.34
FGFR1 P11362 1/20 0.34
PDGFRA P16234 1/20 0.34
PRKACA P17612 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR4 P22455 1/20 0.34
FGFR3 P22607 1/20 0.34
PRKACG P22612 1/20 0.34
PRKACB P22694 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650754 0.91 CDK4 (0.51) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650761 0.90 CDK4 (0.51) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650552 0.85 CDK4 (0.53) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650757 0.85 CDK4 (0.35) CDK4CCND1CDK6CDK2CCNT1
SCHEMBL22650556 0.82 CDK4 (0.52) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650551 0.81 CDK6 (0.52) CDK4CCND1CDK6NPC1RAB9A
SCHEMBL22650544 0.77 CDK4 (0.56) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650545 0.75 CDK4 (0.55) CDK4CCND1CDK6BMPR2NPC1
SCHEMBL22650762 0.73 CDK6 (0.67) CDK4CCND1CDK6CDK2CCNT1
SCHEMBL22650749 0.69 CDK4 (0.54) CDK4CCND1CDK6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed