SCHEMBL22650623

SCHEMBL22650623

Cc1nc2c(F)nc(-c3ccnc(Nc4ccc(S(N)(=O)=O)cc4)n3)cc2n1C(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.52
IKBKB O14920 6/20 0.51
GSK3B P49841 3/20 0.51
DKK1 O94907 2/20 0.51
CDK4 P11802 6/20 0.51
CDK1 P06493 4/20 0.51
CCNB1 P14635 4/20 0.51
CCNT1 O60563 3/20 0.51
CDK9 P50750 3/20 0.51
MAPK8 P45983 2/20 0.51
CCNA2 P20248 2/20 0.51
CDK7 P50613 2/20 0.51
CCNH P51946 2/20 0.51
CCNA1 P78396 2/20 0.51
CCNE1 P24864 2/20 0.51
CCND1 P24385 2/20 0.51
CSNK2A2 P19784 1/20 0.51
CCND3 P30281 1/20 0.51
MAPK9 P45984 1/20 0.51
CSNK1A1 P48729 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650537 0.84 CDK2 (0.50) CDK2IKBKBGSK3BDKK1CDK4
SCHEMBL6605944 0.79 CDK2 (0.60) CDK2IKBKBGSK3BDKK1CDK4
SCHEMBL4822550 0.79 CDK2 (0.63) CDK2IKBKBGSK3BDKK1CDK4
SCHEMBL22650625 0.75 EGFR (0.43) CDK2CDK4CDK1CCNB1CCND1
SCHEMBL22650362 0.74 CDK4 (0.36) CDK2CDK4CDK1CCNB1CDK9
SCHEMBL22650575 0.71 CDK4 (0.57) CDK2CDK4CDK1CCNB1CCNT1
SCHEMBL29491163 0.70 CDK4 (0.46) CDK2GSK3BCDK4CDK1CCNB1
SCHEMBL22650886 0.70 CDK4 (0.46) CDK2GSK3BCDK4CDK1CCNB1
SCHEMBL22650780 0.69 CDK4 (0.54) CDK2CDK4CDK1CCNB1CCNT1
SCHEMBL3524241 0.69 IKBKB (0.61) CDK2IKBKBGSK3BDKK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed