SCHEMBL22650629

SCHEMBL22650629

COc1nc(-c2nc(Nc3ccc(N4CCN(CCF)CC4=O)cn3)ncc2F)cc2c1ncn2C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 20/20 0.41
CDK4 P11802 9/20 0.41
CDK1 P06493 7/20 0.41
CDK2 P24941 5/20 0.41
CCNB1 P14635 3/20 0.41
CCNE1 P24864 3/20 0.41
CCND1 P24385 8/20 0.38
CCNA2 P20248 5/20 0.38
CCND3 P30281 5/20 0.38
CSF1R P07333 1/20 0.38
CDK7 P50613 2/20 0.37
CDK9 P50750 2/20 0.37
CCNE2 O96020 3/20 0.37
CIT O14578 1/20 0.37
GAK O14976 1/20 0.37
DYRK3 O43781 1/20 0.37
CCNT1 O60563 1/20 0.37
STK16 O75716 1/20 0.37
CCNK O75909 1/20 0.37
STK10 O94804 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650547 0.93 CDK6 (0.43) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650560 0.89 CCND1 (0.36) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650558 0.89 CDK6 (0.47) CDK6CDK4CDK1CDK2CCNE1
SCHEMBL22650949 0.86 CDK6 (0.45) CDK6CDK4CDK1CDK2CCND1
SCHEMBL22650550 0.85 CDK4 (0.42) CDK6CDK4CDK1CDK2CCND1
SCHEMBL22650452 0.82 CDK4 (0.54) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650952 0.82 CDK4 (0.49) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650429 0.81 CCND1 (0.40) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650557 0.80 CDK4 (0.53) CDK6CDK4CDK1CDK2CCNB1
SCHEMBL22650956 0.79 CDK6 (0.59) CDK6CDK4CDK1CDK2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed