SCHEMBL22650749

SCHEMBL22650749

CC(C)n1cnc2c1CN(c1nc(Cl)ncc1F)CC2

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.54
CCND1 P24385 2/20 0.54
CDK6 Q00534 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.49
MAPT P10636 1/20 0.43
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
RPS6KA5 O75582 1/20 0.32
PDE10A Q9Y233 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ABL1 P00519 3/20 0.31
BCR P11274 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650742 0.77 TRPV1 (0.40) CDK4CCND1CDK6
SCHEMBL18081432 0.75 CDK6 (0.55) CDK4CCND1CDK6SMN1; SMN2MAPT
SCHEMBL22650762 0.73 CDK6 (0.67) CDK4CCND1CDK6
SCHEMBL22650544 0.73 CDK4 (0.56) CDK4CCND1CDK6SMN1; SMN2
SCHEMBL22650545 0.72 CDK4 (0.55) CDK4CCND1CDK6SMN1; SMN2
SCHEMBL22650555 0.71 CDK6 (1.00) CDK4CCND1CDK6
SCHEMBL22650552 0.70 CDK4 (0.53) CDK4CCND1CDK6SMN1; SMN2
SCHEMBL18081435 0.70 MAPT (0.53) CDK4CCND1CDK6SMN1; SMN2MAPT
SCHEMBL19773558 0.69 SMN1; SMN2 (0.45) CDK4CCND1CDK6SMN1; SMN2MAPT
SCHEMBL24817958 0.68 CDK4 (0.35) CDK4CCND1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed