SCHEMBL22650828

SCHEMBL22650828

COc1nc(-c2nc(Cl)ncc2C)cc2c1nc(C)n2C(C)C

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 13/20 0.33
CDK6 Q00534 10/20 0.33
CCND1 P24385 5/20 0.33
CCND3 P30281 4/20 0.33
EGFR P00533 3/20 0.33
CDK1 P06493 7/20 0.32
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
MDM2 Q00987 3/20 0.31
CDK2 P24941 1/20 0.31
CCNB1 P14635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650829 0.91 CDK4 (0.34) CDK4CDK6CCND1CCND3EGFR
SCHEMBL22650586 0.89 EGFR (0.39) CDK4CDK6CCND1CCND3EGFR
SCHEMBL22650827 0.81 CDK4 (0.39) CDK4CDK6CCND1CCND3EGFR
SCHEMBL22650358 0.78 EGFR (0.33) CDK4CDK6CCND1CCND3EGFR
SCHEMBL22650743 0.76 DAPK1 (0.33) CDK4CCND1EGFRCDK1PDE1A
SCHEMBL29491180 0.76 DAPK1 (0.33) CDK4CCND1EGFRCDK1PDE1A
SCHEMBL22650826 0.76 AAK1 (0.38) CDK4CDK6CCND1CCND3EGFR
SCHEMBL19836272 0.74 CDK4 (0.51) CDK4CDK6CCND1CCND3EGFR
SCHEMBL20987199 0.71 CDK4 (0.53) CDK4CDK6CCND1CCND3EGFR
SCHEMBL30309451 0.71 CDK4 (0.53) CDK4CDK6CCND1CCND3EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed