SCHEMBL22650844

SCHEMBL22650844

Cc1nc(N)ccc1C(=O)N1CCC(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.54
MERTK Q12866 1/20 0.48
NAMPT P43490 1/20 0.48
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
CFTR P13569 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
AKT1 P31749 1/20 0.41
KCNA3 P22001 1/20 0.41
MAP4K4 O95819 2/20 0.41
MCL1 Q07820 1/20 0.41
CTSK P43235 2/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15252462 0.83 CKS1B (0.52) PARP1CKS1BSKP1SKP2KCNA3
SCHEMBL18918808 0.81 PARP1 (0.57) PARP1MERTKNAMPTCKS1BSKP1
SCHEMBL22650456 0.81 GABRP (0.48) PARP1GABRPGABRDGABRA1GABRB1
SCHEMBL30657804 0.80 PARP1 (0.57) PARP1MERTKNAMPTCKS1BSKP1
SCHEMBL31267085 0.79 PARP1 (0.53) PARP1MERTKNAMPTCFTRHDAC3
SCHEMBL4700826 0.79 PARP1 (0.50) PARP1MERTKNAMPTCKS1BSKP1
SCHEMBL29979363 0.78 NAMPT (0.65) PARP1NAMPTCFTRHDAC3HDAC1
SCHEMBL22650451 0.77 PARP1 (0.44) PARP1MERTKNAMPTCKS1BSKP1
SCHEMBL12644375 0.77 NAMPT (0.70) PARP1NAMPTCKS1BSKP1SKP2
SCHEMBL29268404 0.77 NPC1 (0.49) PARP1MERTKNAMPTCFTRMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed