SCHEMBL2265323

SCHEMBL2265323

CCN(CC)C(=O)c1c(-c2ccc(F)cc2)nc(Cc2ccc(S(=O)(=O)O)cc2)nc1C(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.42
GCGR P47871 1/20 0.34
RECQL P46063 1/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
PTGS1 P23219 2/20 0.33
TSPO P30536 1/20 0.33
ABCC3 O15438 1/20 0.33
ABCC4 O15439 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
PDE6D O43924 1/20 0.33
NR1I2 O75469 1/20 0.33
HMGCR P04035 1/20 0.33
PDE4D Q08499 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2221508 0.79 GCGR (0.41) GCGRRECQLTSPOALDH1A1
SCHEMBL2222001 0.75 HMGCR (0.54) ABCC3ABCC4ALDH1A1CYP3A4PDE6D
SCHEMBL2222044 0.75 PTGS2 (0.38) PTGS2GCGRRECQLTSPOABCC3
SCHEMBL778955 0.65 EGFR (0.47) HTR2AALDH1A1
SCHEMBL28301018 0.64 GCGR (0.41) GCGRHMGCR
SCHEMBL8199366 0.64 ALDH1A1 (0.44) PTGS2GCGRALDH1A1
SCHEMBL10153184 0.63 GCGR (0.43) GCGR
SCHEMBL29038363 0.62 GCGR (0.55) PTGS2GCGRPTGS1ALDH1A1CYP3A4
SCHEMBL14248583 0.62 GCGR (0.43) GCGRALDH1A1
SCHEMBL28300691 0.62 PTGS2 (0.42) PTGS2GCGRPTGS1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083495-A2 PROCESS FOR THE PREPARATION OF DIHYDROXY PROTECTED DERIVATIVES AND NOVEL INTERMEDIATE COMPOUNDS MSN LABORATORIES LIMITED (IN) 2011-07-14 WO claimed