SCHEMBL22667253

SCHEMBL22667253

COc1c(O)cc(O)c2c(=O)cc(-c3ccc(N4CCN(CCO)CC4)cc3)oc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP8 P40818 11/20 1.00
CCNT1 O60563 5/20 0.65
CDK9 P50750 5/20 0.65
PARP1 P09874 3/20 0.60
PARP2 Q9UGN5 3/20 0.60
CCNA2 P20248 3/20 0.59
CDK2 P24941 3/20 0.59
GABRP O00591 1/20 0.59
GABRD O14764 1/20 0.59
KDM1A O60341 1/20 0.59
PKM P14618 1/20 0.59
GABRA1 P14867 1/20 0.59
GABRB1 P18505 1/20 0.59
GABRG2 P18507 1/20 0.59
CCNC P24863 1/20 0.59
GABRB3 P28472 1/20 0.59
GABRA5 P31644 1/20 0.59
GABRA3 P34903 1/20 0.59
PTGS2 P35354 1/20 0.59
GABRA2 P47869 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22667248 0.89 USP8 (1.00) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL28953790 0.87 USP8 (1.00) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL22667264 0.84 USP8 (1.00) USP8CCNT1CDK9PARP1PARP2
SCHEMBL22667252 0.84 USP8 (0.92) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL22667238 0.78 CCNT1 (1.00) USP8CCNT1CDK9PARP1PARP2
4'-Hydroxywogonin SCHEMBL29455103 0.78 GABRP (0.81) USP8CCNT1CDK9CCNA2CDK2
4'-Hydroxywogonin SCHEMBL738981 0.78 GABRP (0.81) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL22667243 0.77 USP8 (0.77) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL22667251 0.77 USP8 (0.81) USP8CCNT1CDK9CCNA2CDK2
SCHEMBL22667241 0.76 CCNT1 (0.82) USP8CCNT1CDK9CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228513-A1 NOVEL CDK9 INHIBITOR BASED ON BENZOPYRAN STRUCTURE, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2020-11-19 WO disclosed