SCHEMBL22667448

SCHEMBL22667448

COc1c(OCc2ccccc2)cc(O)c2c(=O)cc(-c3cccc(N4CCOCC4)c3)oc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP8 P40818 7/20 0.60
ACHE P22303 1/20 0.56
PLK1 P53350 1/20 0.56
BACE1 P56817 1/20 0.56
CYP1A1 P04798 2/20 0.54
CYP1B1 Q16678 2/20 0.54
CDK2 P24941 2/20 0.51
CDK9 P50750 2/20 0.51
GABRP O00591 1/20 0.51
GABRD O14764 1/20 0.51
KDM1A O60341 1/20 0.51
CCNT1 O60563 1/20 0.51
PKM P14618 1/20 0.51
GABRA1 P14867 1/20 0.51
GABRB1 P18505 1/20 0.51
GABRG2 P18507 1/20 0.51
CCNA2 P20248 1/20 0.51
CCNC P24863 1/20 0.51
GABRB3 P28472 1/20 0.51
GABRA5 P31644 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28848511 0.86 USP8 (0.70) USP8ACHEPLK1BACE1CDK2
SCHEMBL22667251 0.85 USP8 (0.81) USP8ACHEPLK1BACE1CYP1A1
SCHEMBL21335354 0.85 ACHE (0.77) ACHEPLK1BACE1CDK2CDK9
SCHEMBL22667447 0.83 ACHE (0.64) ACHEPLK1BACE1CYP1A1CDK2
SCHEMBL28848659 0.79 ACHE (0.67) ACHEPLK1BACE1CYP1A1CYP1B1
Moslosooflavone SCHEMBL29822243 0.74 ACHE (1.00) ACHEPLK1BACE1CDK2CDK9
Moslosooflavone SCHEMBL6070206 0.74 ACHE (1.00) ACHEPLK1BACE1CDK2CDK9
SCHEMBL22667444 0.73 ABCB1 (0.54) ACHEPLK1BACE1CYP1A1CYP1B1
SCHEMBL25301059 0.73 ABCB1 (0.65) ACHEPLK1BACE1CYP1A1CYP1B1
SCHEMBL29588215 0.72 ACHE (0.65) USP8ACHEPLK1BACE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228513-A1 NOVEL CDK9 INHIBITOR BASED ON BENZOPYRAN STRUCTURE, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2020-11-19 WO disclosed