SCHEMBL22667997

SCHEMBL22667997

Nc1ccnn1-c1cccc2cnncc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.44
CYP3A4 P08684 3/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 3/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 4/20 0.32
TP53 P04637 3/20 0.32
MAPT P10636 3/20 0.32
MEN1 O00255 2/20 0.32
HPGD P15428 2/20 0.32
ALOX15 P16050 2/20 0.32
CASP1 P29466 2/20 0.32
KMT2A Q03164 2/20 0.32
HSD17B10 Q99714 2/20 0.32
APAF1 O14727 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818549 0.83 POLB (0.52) POLBCYP3A4LMNACYP1A2CYP2D6
SCHEMBL15209780 0.72 SLC9A1 (0.46) POLBCYP3A4LMNAKDM4EMAPT
SCHEMBL4753091 0.69 POLB (0.47) POLB
SCHEMBL544410 0.68 POLB (0.55) POLBMEN1HPGDKMT2ASMN1; SMN2
SCHEMBL15428731 0.68 POLB (0.55) POLBALDH1A1KDM4EPKM
SCHEMBL10992734 0.68 POLB (0.55) POLBALDH1A1KDM4ETP53PKM
SCHEMBL1816971 0.68 POLB (0.55) POLBLMNAALDH1A1TP53MAPT
SCHEMBL659324 0.68 CYP3A4 (0.57) POLBCYP3A4LMNACYP1A2CYP2D6
SCHEMBL31586389 0.68 CYP3A4 (0.57) POLBCYP3A4LMNACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL11473793 0.67 POLB (0.53) POLBALDH1A1KDM4ETP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3738958-A1 AZA-ARYL 1H-PYRAZOL-1-YL BENZENE SULFONAMIDES AS CCR(9) ANTAGONISTS ChemoCentryx, Inc. (US) 2020-11-18 EP disclosed