SCHEMBL22669019

SCHEMBL22669019

FC(F)(F)c1ccccc1N1CCCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.54
TTR P02766 1/20 0.51
HSD11B1 P28845 2/20 0.49
KEAP1 Q14145 1/20 0.48
HTR1A P08908 1/20 0.48
TRPV1 Q8NER1 3/20 0.48
MAPK1 P28482 2/20 0.47
RBP4 P02753 1/20 0.46
DRD4 P21917 1/20 0.46
GRM2 Q14416 1/20 0.46
NOTUM Q6P988 3/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27647544 0.98 AKR1C3 (0.53) AKR1C3TTRHSD11B1KEAP1HTR1A
SCHEMBL23211918 0.96 AKR1C3 (0.54) AKR1C3TTRHSD11B1KEAP1HTR1A
SCHEMBL30407607 0.96 AKR1C3 (0.54) AKR1C3TTRHSD11B1KEAP1HTR1A
SCHEMBL4064652 0.84 AKR1C3 (0.51) AKR1C3TTRHSD11B1HTR1ATRPV1
Tert-Butyl Formate SCHEMBL27869235 0.83 HSD11B1 (0.47) AKR1C3TTRHSD11B1KEAP1HTR1A
SCHEMBL7624363 0.82 ADRA2C (0.55) AKR1C3TTRHSD11B1HTR1ATRPV1
SCHEMBL231778 0.82 EPHX2 (0.61) AKR1C3HTR1AALDH1A1LMNACYP1A2
SCHEMBL20752166 0.82 AKR1C3 (0.70) AKR1C3TTRHSD11B1HTR1ANOTUM
SCHEMBL2299021 0.82 AKR1C3 (0.50) AKR1C3TTRHSD11B1HTR1ATRPV1
SCHEMBL31096264 0.82 ADRA2C (0.55) AKR1C3TTRHSD11B1HTR1ATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020229968-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF ALECTOS THERAPEUTICS INC. (CA) 2020-11-19 WO disclosed
CN-109496213-A Spiro-compound and its preparation and application 阿比德治疗公司 2019-03-19 CN disclosed