SCHEMBL22677334

SCHEMBL22677334

COC(=O)c1ncnc2c1CCN2

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NNMT P40261 3/20 0.46
NPSR1 Q6W5P4 1/20 0.37
DRD1 P21728 2/20 0.36
MKNK1 Q9BUB5 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PARP1 P09874 1/20 0.34
RET P07949 1/20 0.33
KDM4E B2RXH2 2/20 0.33
STAT3 P40763 1/20 0.33
HIF1A Q16665 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
EGFR P00533 1/20 0.32
ERBB2 P04626 1/20 0.32
KDR P35968 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12775966 0.79 AKT1 (0.37) NPSR1L3MBTL1PARP1KDM4ESTAT3
SCHEMBL17541159 0.79 NNMT (0.60) NNMTDRD1MKNK1RETKDR
SCHEMBL12590774 0.77 SPR (0.39) NPSR1PARP1KDM4EALDH1A1
SCHEMBL14320242 0.75 NNMT (0.46) NNMTPARP1KDM4EKDM4CALDH1A1
SCHEMBL12590744 0.74 PRKACA (0.41) NPSR1L3MBTL1PARP1KDM4ESTAT3
SCHEMBL27879194 0.73 NPSR1 (0.35) NPSR1L3MBTL1KDM4ESTAT3HIF1A
SCHEMBL2600057 0.71 DRD1 (0.49) NNMTDRD1MKNK1RETKDR
SCHEMBL12776648 0.71 ENPP1 (0.44) KDM4EALDH1A1
SCHEMBL3507179 0.69 EGFR (0.44) NNMTDRD1RETEGFRERBB2
SCHEMBL3506856 0.69 EGFR (0.49) NNMTRETEGFRERBB2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020231990-A1 FGFR INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2020-11-19 WO disclosed