SCHEMBL22681817

SCHEMBL22681817

Cc1ccc(N(C)c2ccc3c(c2)CCC3)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
LMNA P02545 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
THRB P10828 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
POLB P06746 2/20 0.45
MAPT P10636 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TSHR P16473 1/20 0.40
RAPGEF4 Q8WZA2 1/20 0.40
DPP4 P27487 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13569439 0.96 ALDH1A1 (0.43) ALDH1A1LMNASMN1; SMN2THRBL3MBTL1
SCHEMBL22681798 0.87 RXRA (0.43) ALDH1A1LMNASMN1; SMN2THRBL3MBTL1
SCHEMBL22681601 0.85 RXRA (0.46) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL22681604 0.84 NPC1 (0.46) ALDH1A1LMNASMN1; SMN2THRBL3MBTL1
SCHEMBL22682009 0.83 RXRA (0.43) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL19049725 0.82 RXRA (0.39) ALDH1A1MAPTRXRARXRBRXRG
SCHEMBL17378763 0.81 RXRA (0.46) ALDH1A1LMNASMN1; SMN2MAPTRXRA
SCHEMBL22681835 0.81 ALDH1A1 (0.50) ALDH1A1L3MBTL1NPC1RAB9APOLB
SCHEMBL22681707 0.81 NPC1 (0.42) ALDH1A1SMN1; SMN2NPC1RAB9APOLB
SCHEMBL22682095 0.81 RXRA (0.49) LMNAL3MBTL1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160952-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2020-12-02 EP disclosed
EP-3741749-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-25 EP disclosed
EP-3738960-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-18 EP disclosed