SCHEMBL22685172

SCHEMBL22685172

C#Cc1ccc(C(=O)NC2(c3ccc(-c4ccc(F)cn4)cc3)CCC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.44
PTPN6 P29350 1/20 0.44
PTPN11 Q06124 1/20 0.44
NPC1 O15118 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HDAC2 Q92769 5/20 0.40
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
CNR2 P34972 1/20 0.39
P2RX7 Q99572 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
AKT1 P31749 1/20 0.37
MCHR1 Q99705 2/20 0.37
PRKAA2 P54646 1/20 0.37
BTK Q06187 1/20 0.36
DGAT1 O75907 1/20 0.35
PDE2A O00408 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22685161 0.96 PTPN1 (0.46) PTPN1PTPN6PTPN11NPC1RXFP1
SCHEMBL22685168 0.85 PTPN1 (0.40) PTPN1PTPN6PTPN11NPC1RXFP1
SCHEMBL22684819 0.84 PTPN1 (0.42) PTPN1PTPN6PTPN11NPC1RXFP1
SCHEMBL22685160 0.83 WDR91 (0.41) PTPN1PTPN6PTPN11HDAC2HDAC3
SCHEMBL22657405 0.78 WDR91 (0.39) PTPN1PTPN6PTPN11HDAC2HDAC3
SCHEMBL22685095 0.75 MCHR1 (0.39) NPC1CNR2CTSLCTSBCTSS
SCHEMBL28547259 0.75 NPC1 (0.44) PTPN1PTPN6PTPN11NPC1RXFP1
SCHEMBL22685186 0.75 PTPN1 (0.48) PTPN1PTPN6PTPN11NPC1RXFP1
SCHEMBL22657410 0.74 WDR91 (0.40) NPC1HDAC2HDAC3HDAC1HDAC6
SCHEMBL22657417 0.74 MKNK1 (0.45) HDAC1HDAC6CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228823-A1 NOVEL AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2020-11-19 WO disclosed