SCHEMBL22702016

SCHEMBL22702016

CC(C)(C)C(O)c1cccc(N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.44
CASP1 P29466 1/20 0.44
RECQL P46063 1/20 0.44
CPN1 P15169 1/20 0.43
CPB2 Q96IY4 1/20 0.43
ALDH1A1 P00352 5/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
CA12 O43570 1/20 0.41
CA7 P43166 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA14 Q9ULX7 1/20 0.41
SLC6A2 P23975 4/20 0.41
SLC6A4 P31645 4/20 0.41
SLC6A3 Q01959 4/20 0.41
CYP2D6 P10635 3/20 0.41
KCNH2 Q12809 2/20 0.41
ADRB1 P08588 2/20 0.40
AOC3 Q16853 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21525433 0.88 CYP3A4 (0.44) CYP3A4CASP1RECQLCPN1CPB2
SCHEMBL10415544 0.79 ACP3 (0.44) ALDH1A1TDP1ADRB1AOC3MIF
SCHEMBL14443273 0.79 ADRB1 (0.58) CYP3A4ALDH1A1CA2CA9CA12
SCHEMBL4282395 0.79 TSHR (0.47) CYP3A4CASP1RECQLCPN1CPB2
SCHEMBL30317737 0.79 ADRB1 (0.58) CYP3A4ALDH1A1CA2CA9CA12
SCHEMBL19589404 0.78 HDAC8 (0.44) CYP3A4ALDH1A1TDP1ADRB1AOC3
SCHEMBL12791279 0.78 ACP3 (0.43) SLC6A2SLC6A4SLC6A3KCNH2ADRB1
SCHEMBL1525214 0.78 SLC6A2 (0.42) CYP3A4ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL5378913 0.78 CES2 (0.47) SLC6A2SLC6A4AOC3
SCHEMBL26262585 0.78 ACP3 (0.43) SLC6A2SLC6A4SLC6A3KCNH2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3319955-B1 6-AMINO-QUINOLINE-3-CARBONITRILS AS COT MODULATORS GILEAD SCIENCES INC (US) 2020-11-25 EP disclosed