SCHEMBL22705448

SCHEMBL22705448

Cc1noc([C@@H]2CCCN2C(O)C(C)(C)Sc2ccc(Cl)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
ENPP2 Q13822 2/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
HDAC1 Q13547 3/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC5 Q9UQL6 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22705654 0.80 HCRTR1 (0.44) SMN1; SMN2MAPTLMNAENPP2HCRTR1
SCHEMBL22705498 0.78 ENPP2 (0.38) HDAC6SMN1; SMN2MAPTLMNAENPP2
SCHEMBL22705449 0.76 ENPP2 (0.38) HDAC6ENPP2HCRTR1HCRTR2HDAC1
SCHEMBL12890751 0.70 CHRM2 (0.43) HDAC6HDAC1HDAC8HDAC5
SCHEMBL24597834 0.69 HDAC6 (0.39) HDAC6HCRTR1HCRTR2HDAC1HDAC8
SCHEMBL24597827 0.68 HCRTR1 (0.46) SMN1; SMN2MAPTLMNAENPP2HCRTR1
SCHEMBL22705500 0.68 HCRTR1 (0.46) SMN1; SMN2MAPTLMNAENPP2HCRTR1
SCHEMBL22705433 0.68 LMNA (0.47) MAPTLMNAENPP2HCRTR1HCRTR2
SCHEMBL9963155 0.67 HDAC6 (0.43) HDAC6HDAC1HDAC8HDAC5
SCHEMBL22705454 0.65 CPT1A (0.44) ENPP2HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020233618-A1 INHIBITORS FOR PROGRAMMED CELL NECROSIS AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海有机化学研究所 (CN) 2020-11-26 WO disclosed