SCHEMBL2271014

SCHEMBL2271014

CN1CCCC(NC(=O)CC2CCN(c3ncc(C#N)cc3NC(=O)c3cccc(Cl)c3)CC2)C1.N#Cc1cnc(N2CCC(CC(=O)Nc3cccnc3)CC2)c(NC(=O)c2cccc(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.55
GRM5 P41594 3/20 0.42
GPR6 P46095 11/20 0.42
USP30 Q70CQ3 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
BTK Q06187 2/20 0.38
BRAF P15056 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2271430 0.93 CXCR3 (0.48) CXCR3GRM5GPR6MEN1KMT2A
SCHEMBL2269616 0.91 CXCR3 (0.65) CXCR3GPR6USP30MEN1KMT2A
SCHEMBL2268315 0.84 CXCR3 (0.57) CXCR3GRM5MEN1KMT2ABTK
SCHEMBL2270608 0.84 CXCR3 (0.57) CXCR3GRM5MEN1KMT2ABTK
SCHEMBL2267846 0.84 CXCR3 (0.54) CXCR3GRM5MEN1KMT2ABTK
SCHEMBL2362900 0.84 CCR2 (0.46) GPR6BTK
SCHEMBL2221638 0.82 CXCR3 (0.78) CXCR3GRM5USP30MEN1KMT2A
SCHEMBL2223197 0.81 CXCR3 (0.48) CXCR3GRM5MEN1KMT2ABTK
SCHEMBL2264590 0.79 CXCR3 (0.53) CXCR3GPR6MEN1KMT2A
SCHEMBL2269437 0.79 CXCR3 (0.48) CXCR3GPR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084985-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-14 WO disclosed