SCHEMBL22720186

SCHEMBL22720186

Nc1cc(F)c(F)cc1C(=O)Nc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
TDP1 Q9NUW8 2/20 0.54
ALDH1A1 P00352 1/20 0.51
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
NCOR2 Q9Y618 1/20 0.51
FADS1 O60427 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
LMNA P02545 2/20 0.50
TP53 P04637 2/20 0.50
HPGD P15428 2/20 0.50
KDM4E B2RXH2 1/20 0.50
HTT P42858 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PRKCI P41743 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13362653 0.87 MEN1 (0.53) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL6590611 0.84 NPC1 (0.58) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL13162555 0.82 CYP11B2 (0.77) MEN1KMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL10430505 0.82 FADS1 (0.56) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL12885792 0.82 FADS1 (0.72) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL5668526 0.81 PTGS1 (0.71) MEN1KMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL5224168 0.80 GCK (0.60) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL7630470 0.79 KMT2A (0.57) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL6812861 0.79 MEN1 (0.58) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL734813 0.78 CYP1A2 (0.59) MEN1KMT2ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
CN-110041272-B 2- (2-chlorphenyl) quinazoline-4 (3H) -ketone derivative and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-30 CN disclosed
CN-110041273-B 2- (2-chloro-4-methylphenyl) quinazoline-4 (3H) -ketone compound and medical application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-20 CN disclosed
CN-110041273-A 2- (the chloro- 4- aminomethyl phenyl of 2-) quinazoline -4 (3H) -one class compound and its medical usage 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed
CN-110041272-A 2- (2- chlorphenyl) quinazoline -4 (3H) -one analog derivative and its preparation method and application 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed