SCHEMBL22720253

SCHEMBL22720253

Cc1nc(Cl)nc(N2CCN(C(=O)OC(C)(C)C)CC2)c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
POLB P06746 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
CKS1B P61024 1/20 0.41
SKP1 P63208 1/20 0.41
SKP2 Q13309 1/20 0.41
GBA1 P04062 2/20 0.41
MAPT P10636 2/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TLR9 Q9NR96 1/20 0.40
BACE1 P56817 1/20 0.40
SUV39H2 Q9H5I1 1/20 0.39
MAP4K4 O95819 1/20 0.39
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720236 0.84 TLR9 (0.44) KCNH2CNR1CNR2MEN1KMT2A
SCHEMBL20011912 0.82 POLB (0.47) CNR1CNR2POLBMEN1KMT2A
SCHEMBL30060994 0.82 POLB (0.47) CNR1CNR2POLBMEN1KMT2A
SCHEMBL28768664 0.81 MAPT (0.50) KCNH2CNR1CNR2POLBMEN1
SCHEMBL29673158 0.81 MAPT (0.50) KCNH2CNR1CNR2POLBMEN1
SCHEMBL28646478 0.78 KCNH2 (0.39) KCNH2CNR1CNR2POLBMEN1
SCHEMBL15413007 0.78 CKS1B (0.48) CNR1CNR2POLBMEN1KMT2A
SCHEMBL19995252 0.78 TLR9 (0.44) CNR1CNR2POLBMEN1KMT2A
SCHEMBL30061006 0.78 TLR9 (0.44) CNR1CNR2POLBMEN1KMT2A
SCHEMBL29421769 0.78 CKS1B (0.48) CNR1CNR2POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-112552294-B Piperazine heterocyclic derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-19 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
CN-112552294-A Piperazine heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed