SCHEMBL22720236

SCHEMBL22720236

COc1nc(C)c(Br)c(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.44
KCNH2 Q12809 2/20 0.41
SMPD3 Q9NY59 2/20 0.41
GBA1 P04062 2/20 0.40
CKS1B P61024 2/20 0.40
SKP1 P63208 2/20 0.40
SKP2 Q13309 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.39
SUV39H2 Q9H5I1 1/20 0.39
MAP4K4 O95819 1/20 0.39
KIT P10721 1/20 0.39
TLR7 Q9NYK1 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
USP2 O75604 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22724587 0.85 TLR9 (0.44) TLR9SMPD3GBA1CKS1BSKP1
SCHEMBL22720253 0.84 KCNH2 (0.42) TLR9KCNH2GBA1CKS1BSKP1
SCHEMBL22720228 0.83 TLR9 (0.42) TLR9SMPD3GBA1CKS1BSKP1
SCHEMBL22720285 0.79 KRAS (0.42) KCNH2
SCHEMBL22720279 0.78 TLR9 (0.43) TLR9SMPD3GBA1CKS1BSKP1
SCHEMBL21734104 0.76 GBA1 (0.44) TLR9GBA1CKS1BSKP1SKP2
SCHEMBL18133895 0.76 TLR9 (0.45) TLR9KCNH2GBA1SUV39H2MAP4K4
SCHEMBL16637413 0.75 TLR9 (0.53) TLR9KCNH2GBA1SUV39H2KIT
SCHEMBL22873609 0.74 GPR119 (0.55) TLR9SMPD3GBA1CKS1BSKP1
SCHEMBL31652099 0.74 TLR9 (0.54) TLR9SMPD3GBA1CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-112552294-B Piperazine heterocyclic derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-19 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
CN-112552294-A Piperazine heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed