SCHEMBL22720277

SCHEMBL22720277

CN1CCCC1COc1nc2c(c(N3CCN(C(=O)O)C(C(C)(C)C)C3)n1)CCC2

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.49
VHL P40337 1/20 0.44
CDK7 P50613 1/20 0.44
CCNH P51946 1/20 0.44
MNAT1 P51948 1/20 0.44
SOS1 Q07889 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692005 0.85 KRAS (0.55) KRAS
SCHEMBL28692003 0.85 KRAS (0.55) KRAS
SCHEMBL22720289 0.83 KRAS (0.40) KRASSOS1
SCHEMBL22720275 0.82 KRAS (0.43) KRASSOS1
SCHEMBL22720273 0.80 KRAS (0.52) KRAS
SCHEMBL22724649 0.80 KRAS (0.52) KRAS
SCHEMBL25349824 0.78 KRAS (0.47) KRASVHLCDK7CCNHMNAT1
SCHEMBL25349832 0.78 KRAS (0.47) KRASVHLCDK7CCNHMNAT1
SCHEMBL21722155 0.78 KRAS (0.52) KRAS
SCHEMBL22720270 0.77 KRAS (0.37) KRASSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed