SCHEMBL22726316

SCHEMBL22726316

C=C(CCC)C(CC)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.40
PDE2A O00408 2/20 0.38
CYP2C9 P11712 6/20 0.37
CYP1A2 P05177 5/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 5/20 0.37
CYP2C19 P33261 5/20 0.37
TP53 P04637 3/20 0.37
CYP2D6 P10635 2/20 0.37
HRH3 Q9Y5N1 3/20 0.36
MC4R P32245 1/20 0.36
SLC6A4 P31645 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1903665 0.75 AKR1C3 (0.59) CYP3A4CYP2C9CYP1A2MEN1KMT2A
SCHEMBL11444719 0.73 CES2 (0.45) CYP3A4PDE2ACYP2C9CYP1A2MEN1
Hydrochloric Acid SCHEMBL2763475 0.73 AKR1C3 (0.58) CYP3A4CYP2C9CYP1A2MEN1KMT2A
SCHEMBL23892021 0.73 SMN1; SMN2 (0.38) CYP3A4PDE2ACYP2C9CYP1A2MEN1
SCHEMBL26495295 0.73 CYP3A4 (0.42) CYP3A4PDE2ACYP2C9CYP1A2MEN1
SCHEMBL26697470 0.71 PPARG (0.48) CYP3A4CYP2C9CYP1A2MEN1KMT2A
SCHEMBL21573071 0.71 HRH3 (0.37) CYP3A4CYP2C9CYP1A2MEN1KMT2A
SCHEMBL10073359 0.70 PDE2A (0.56) PDE2ACES2CES1
SCHEMBL15387995 0.70 PDE2A (0.56) PDE2ACES2CES1
SCHEMBL478137 0.70 PDE2A (0.56) PDE2ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057950-B1 PHENYL LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T JANSSEN PHARMACEUTICA NV (BE) 2020-12-02 EP disclosed