SCHEMBL2273158

SCHEMBL2273158

COc1ccc(C)c2c1OC[C@H](CCN)Cn1c-2c(C2CCCCC2)c2ccc(C(=O)O)cc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.46
MMP12 P39900 1/20 0.46
NR1I2 O75469 2/20 0.33
SCN9A Q15858 2/20 0.33
CFB P00751 5/20 0.33
KCNH2 Q12809 3/20 0.32
CYP3A4 P08684 2/20 0.32
SCN5A Q14524 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2274159 0.92 PRKCA (0.44) PRKCAMMP12NR1I2SCN9ACFB
SCHEMBL4216548 0.89 PRKCA (0.52) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL2280300 0.88 PRKCA (0.47) PRKCAMMP12NR1I2SCN9ACFB
SCHEMBL2271812 0.87 PRKCA (0.45) PRKCAMMP12NR1I2SCN9ACFB
SCHEMBL2273152 0.82 PRKCA (0.44) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL2276489 0.81 PRKCA (0.40) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL4206439 0.80 PRKCA (0.51) PRKCAMMP12NR1I2SCN9AKCNH2
SCHEMBL2276847 0.79 PRKCA (0.53) PRKCAMMP12NR1I2SCN9ACFB
SCHEMBL2279218 0.77 PRKCA (0.47) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL2273255 0.77 PRKCA (0.54) PRKCAMMP12NR1I2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed