SCHEMBL2273580

SCHEMBL2273580

CCC(c1cnc(-c2cccc(Cc3nn(-c4cnn(C)c4)ccc3=O)c2)nc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.34
MET P08581 1/20 0.32
CTSV O60911 2/20 0.32
CTSL P07711 2/20 0.32
CTSS P25774 2/20 0.32
CTSB P07858 1/20 0.32
CTSK P43235 1/20 0.31
HSD17B13 Q7Z5P4 1/20 0.31
IRAK4 Q9NWZ3 3/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30
IRAK1 P51617 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2220291 0.85 ENPP2 (0.36) ENPP2METCTSVCTSLCTSS
SCHEMBL13275655 0.85 PPARG (0.36) ENPP2METCTSVCTSLCTSS
SCHEMBL13275160 0.83 FYN (0.34) ENPP2METCTSVCTSLCTSS
SCHEMBL2269058 0.83 ENPP2 (0.41) ENPP2METCTSVCTSLCTSS
SCHEMBL2264266 0.82 HSD17B13 (0.37) ENPP2METHSD17B13IRAK4IRAK1
SCHEMBL13275650 0.82 ENPP2 (0.35) ENPP2METCTSVCTSLCTSS
SCHEMBL2273583 0.81 ENPP2 (0.33) ENPP2METCTSVCTSLCTSS
SCHEMBL2219418 0.81 IRAK1 (0.36) ENPP2METCTSVCTSLCTSS
SCHEMBL2271291 0.81 HSD17B13 (0.38) ENPP2METHSD17B13IRAK4IRAK1
SCHEMBL2261414 0.81 HSD17B13 (0.42) ENPP2METHSD17B13IRAK4IRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed