SCHEMBL22738696

SCHEMBL22738696

N=C(N)NCCC[C@@H]1NC(=O)[C@H](CCCCNC(=O)[C@@H](N)CCCCNC(=O)CCCc2ccc(I)cc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CC(=O)O)NC(=O)CNC1=O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.52
ITGAV P06756 8/20 0.52
ITGB1 P05556 2/20 0.52
ITGA5 P08648 2/20 0.52
ITGB5 P18084 5/20 0.51
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
MC4R P32245 7/20 0.45
MC5R P33032 7/20 0.45
MC3R P41968 7/20 0.45
MC1R Q01726 7/20 0.45
CTSG P08311 2/20 0.45
ITGA2B P08514 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23999259 0.94 ITGB3 (0.52) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL7743670 0.91 ITGB3 (0.56) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL22970321 0.91 ITGB3 (0.56) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL19981446 0.91 ITGB3 (0.56) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL7744260 0.91 ITGB3 (0.56) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL22738697 0.88 KEAP1 (0.51) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL22872747 0.86 ITGB3 (0.51) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL7744274 0.85 KEAP1 (0.52) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL20754200 0.84 ITGB3 (0.53) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL24285403 0.84 ITGB3 (0.53) ITGB3ITGAVITGB1ITGA5ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020238800-A1 TARGETED RADIOPHARMACEUTICALS FOR TUMORS, AND COMBINATION THERAPY OF TARGETED RADIOTHERAPY THEREOF AND IMMUNOTHERAPY UNDER GUIDANCE OF IMAGES 北京大学 2020-12-03 WO disclosed