SCHEMBL22758396

SCHEMBL22758396

CCOC(=O)/C(CC(=O)c1cccnc1N)=N\I

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
NAPRT Q6XQN6 1/20 0.42
PRKCI P41743 2/20 0.39
BRD4 O60885 1/20 0.39
P2RX7 Q99572 1/20 0.39
HTT P42858 1/20 0.39
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
HSD17B10 Q99714 1/20 0.37
VCP P55072 2/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
HPGD P15428 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12441324 0.80 NAPRT (0.50) MAPTCYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL13460683 0.77 NAPRT (0.53) MAPTCYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL181049 0.74 ALDH1A1 (0.60) MAPTNAPRTBRD4HTTALDH1A1
SCHEMBL14227406 0.73 NAPRT (0.54) NAPRTPRKCIP2RX7ALDH1A1KDM4E
SCHEMBL13545172 0.72 NAPRT (0.61) MAPTCYP3A4NAPRTPRKCIP2RX7
Hydrochloric Acid SCHEMBL27738327 0.71 NAPRT (0.59) MAPTCYP3A4NAPRTPRKCIP2RX7
SCHEMBL9368829 0.70 NAPRT (0.62) MAPTCYP3A4NAPRTPRKCIP2RX7
SCHEMBL2301544 0.69 HTT (0.45) MAPTCYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL2301534 0.69 HTT (0.45) MAPTCYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL29686396 0.69 PRKCI (0.55) NAPRTPRKCIP2RX7HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020247804-A1 HETEROCYCLE SUBSTITUTED PYRIDINE DERIVATIVE ANTIFUNGAL AGENTS AMPLYX PHARMACEUTICALS, INC. (US) 2020-12-10 WO disclosed