SCHEMBL22759261

SCHEMBL22759261

CC1COCCN1c1nc(Cl)nc(Cl)c1F

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTOR P42345 19/20 0.50
ATR Q13535 1/20 0.40
PIK3CD O00329 1/20 0.38
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
RICTOR Q6R327 1/20 0.38
RPTOR Q8N122 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
MAPKAP1 Q9BPZ7 1/20 0.38
MLST8 Q9BVC4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22759089 1.00 MTOR (0.50) MTORATRPIK3CDPIK3R1PIK3CA
SCHEMBL4974288 0.80 FPR2 (0.37) MTORPIK3R1PIK3CA
SCHEMBL4974284 0.80 FPR2 (0.37) MTORPIK3R1PIK3CA
SCHEMBL24069658 0.79 MTOR (0.44) MTORATRPIK3CDPIK3R1PIK3CA
SCHEMBL3399370 0.78 MTOR (0.44) MTORATRPIK3C3
SCHEMBL3399374 0.78 MTOR (0.44) MTORATRPIK3C3
SCHEMBL2708210 0.77 MTOR (0.47) MTORPIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL2708205 0.77 MTOR (0.47) MTORPIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL2908876 0.76 MTOR (0.41) MTOR
SCHEMBL20692837 0.75 MTOR (0.53) MTORPIK3R1PIK3CARICTORRPTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244613-A1 2, 4, 6-TRI-SUBSTITUTED PYRIMIDINE COMPOUND AS ATR KINASE INHIBITOR 北京泰德制药股份有限公司 2020-12-10 WO disclosed