SCHEMBL22760087

SCHEMBL22760087

CC(C)c1cccc(-n2c(C(=O)O)c(N3CCOCC3)c3c(Cl)c(F)ccc32)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.39
NOTUM Q6P988 2/20 0.39
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
KMO O15229 1/20 0.37
KDM4E B2RXH2 3/20 0.36
HPGD P15428 3/20 0.36
CASP1 P29466 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
NTRK1 P04629 1/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760177 0.90 AKR1C3 (0.44) CYP3A4CYP1A2KMOKDM4EHPGD
SCHEMBL22747901 0.88 HSD17B10 (0.37) KDM4EHPGDALDH1A1LMNATSHR
SCHEMBL22747853 0.88 MAPT (0.42) NOTUMCYP3A4CYP1A2KMOKDM4E
SCHEMBL22748334 0.88 KMO (0.40) NOTUMCYP3A4CYP1A2KMOKDM4E
SCHEMBL22747879 0.86 HPGD (0.42) CYP3A4CYP1A2CYP2C9KMOKDM4E
SCHEMBL22748196 0.86 EDNRA (0.42) NOTUMKMOKDM4EALDH1A1LMNA
SCHEMBL22760131 0.86 KMO (0.39) CYP3A4CYP1A2KMOKDM4EHPGD
SCHEMBL22760212 0.85 NOTUM (0.39) PPARGNOTUMCYP3A4CYP1A2KMO
SCHEMBL22748281 0.85 KMO (0.37) CYP3A4CYP1A2KMOKDM4EHPGD
SCHEMBL22748300 0.85 KMO (0.37) CYP3A4CYP1A2KMOKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed