SCHEMBL22760177

SCHEMBL22760177

O=C(O)c1c(N2CCOCC2)c2c(Cl)c(F)ccc2n1-c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.44
KMO O15229 1/20 0.42
KDM4E B2RXH2 4/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CASP1 P29466 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 6/20 0.40
MAPT P10636 3/20 0.40
TSHR P16473 2/20 0.40
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
PKM P14618 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LMNA P02545 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
EDNRA P25101 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22748334 0.94 KMO (0.40) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22747879 0.93 HPGD (0.42) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22760131 0.92 KMO (0.39) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22747853 0.92 MAPT (0.42) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22747895 0.90 TSHR (0.39) KMOKDM4EHPGDCYP1A2CYP3A4
SCHEMBL22748196 0.90 EDNRA (0.42) KMOKDM4EALDH1A1MAPTTSHR
SCHEMBL22747892 0.90 NOTUM (0.40) KMOKDM4EHPGDCYP1A2CYP3A4
SCHEMBL22760212 0.90 NOTUM (0.39) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22760087 0.90 PPARG (0.39) AKR1C3KMOKDM4EHPGDCYP1A2
SCHEMBL22760100 0.89 SMN1; SMN2 (0.40) KDM4EHPGDALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed