SCHEMBL22760118

SCHEMBL22760118

O=C(O)c1c(N2CCCCC2)c2c(F)c(F)ccc2n1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.38
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
EDNRA P25101 1/20 0.36
LMNA P02545 2/20 0.36
REN P00797 1/20 0.35
MAPT P10636 4/20 0.34
NPC1 O15118 3/20 0.34
TP53 P04637 3/20 0.34
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
TSHR P16473 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ALOX15 P16050 1/20 0.34
STAT1 P42224 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760542 0.88 GAA (0.37) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22760063 0.88 EDNRA (0.39) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22747830 0.88 EDNRA (0.39) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22748355 0.87 EDNRA (0.40) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22760172 0.85 MAPT (0.47) GAAALDH1A1HPGDMEN1KMT2A
SCHEMBL22760100 0.83 SMN1; SMN2 (0.40) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22760499 0.81 NOTUM (0.37) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22747822 0.81 GAA (0.38) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22748265 0.79 HPGD (0.40) GAAALDH1A1HPGDHSD17B10MEN1
SCHEMBL22760495 0.79 FOLH1 (0.37) GAAALDH1A1HPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed