SCHEMBL22760149

SCHEMBL22760149

CCOC(=O)c1c(N2CCOCC2)c2c(Cl)c(F)ccc2n1-c1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.41
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
DGAT1 O75907 1/20 0.39
SOAT1 P35610 1/20 0.39
PIK3CA P42336 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 2/20 0.39
MAPK1 P28482 2/20 0.39
USP2 O75604 1/20 0.39
RECQL P46063 1/20 0.39
HPGD P15428 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760185 0.95 HPGD (0.43) LMNAMAPTDGAT1SOAT1PIK3CA
SCHEMBL22747893 0.93 MAPK1 (0.39) LMNAMAPTSMN1; SMN2KDM4EPIK3CA
SCHEMBL22748357 0.92 JMJD6 (0.39) LMNAMAPTSMN1; SMN2KDM4EDGAT1
SCHEMBL22748253 0.91 HSD17B10 (0.39) LMNAMAPTSMN1; SMN2KDM4EPIK3CA
SCHEMBL22760192 0.91 ALDH1A1 (0.41) LMNAMAPTKDM4EDGAT1SOAT1
SCHEMBL22747825 0.91 HPGD (0.45) LMNAMAPTSMN1; SMN2TP53MAPK1
SCHEMBL22747823 0.91 ALDH1A1 (0.45) LMNAMAPTKDM4EDGAT1SOAT1
SCHEMBL22748239 0.91 HSD17B10 (0.41) LMNAKDM4EPIK3CAHSD17B10TP53
SCHEMBL22760193 0.90 ALDH1A1 (0.45) LMNAMAPTKDM4EPIK3CAHSD17B10
SCHEMBL22747889 0.90 HSD17B10 (0.39) LMNAMAPTSMN1; SMN2KDM4EDGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed