SCHEMBL22760173

SCHEMBL22760173

CCOC(=O)c1c(N)c2c(F)c(F)ccc2n1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
MAPT P10636 5/20 0.53
GAA P10253 3/20 0.53
KDM4E B2RXH2 6/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 3/20 0.48
THRB P10828 2/20 0.46
TP53 P04637 2/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
RECQL P46063 1/20 0.41
ALOX15 P16050 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAT2A P31153 1/20 0.41
HIF1A Q16665 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760094 0.89 ALDH1A1 (0.51) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22747883 0.83 MAPT (0.50) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760172 0.81 MAPT (0.47) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760543 0.80 ALDH1A1 (0.54) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760129 0.76 ALDH1A1 (0.50) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760095 0.75 MAPT (0.48) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760162 0.74 TSHR (0.47) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760544 0.74 MEN1 (0.53) ALDH1A1MAPTGAAKDM4ETHRB
SCHEMBL22748263 0.73 MAPK8 (0.40) ALDH1A1MAPTGAAKDM4EHPGD
SCHEMBL22760117 0.71 FOLH1 (0.36) ALDH1A1MAPTGAAKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed