SCHEMBL2277012

SCHEMBL2277012

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](N(CCOCCO)C(=O)OC(C)(C)C)COc1ccccc1-3

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.56
MMP12 P39900 1/20 0.56
NR1I2 O75469 7/20 0.36
CYP3A4 P08684 3/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 5/20 0.32
SCN5A Q14524 2/20 0.32
CSNK2A1 P68400 1/20 0.31
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2277965 0.94 PRKCA (0.54) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL4212003 0.93 PRKCA (0.65) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2278834 0.92 PRKCA (0.55) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2275101 0.91 PRKCA (0.56) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2276683 0.90 PRKCA (0.52) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2276695 0.88 PRKCA (0.55) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL4208318 0.88 PRKCA (0.62) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2279113 0.87 PRKCA (0.54) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL4210071 0.86 PRKCA (0.62) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2277015 0.84 PRKCA (0.53) PRKCAMMP12NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed