SCHEMBL22787487

SCHEMBL22787487

NNc1c(NC2CC(O)C(CO)C2)ncnc1N[C@@H]1c2ccccc2C[C@@H]1O

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.47
RPS6KB1 P23443 1/20 0.47
NAE1 Q13564 14/20 0.44
UBA3 Q8TBC4 14/20 0.44
SAE1 Q9UBE0 3/20 0.34
UBA2 Q9UBT2 3/20 0.34
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24286184 0.85 NAE1 (0.63) NAE1UBA3SAE1UBA2
SCHEMBL24286013 0.78 SLC29A1 (0.46) NAE1UBA3
SCHEMBL24286025 0.77 NAE1 (0.44) AURKARPS6KB1NAE1UBA3
SCHEMBL22787553 0.76 NAE1 (0.41) NAE1UBA3SAE1UBA2
SCHEMBL22787471 0.76 NAE1 (0.40) AURKARPS6KB1NAE1UBA3
SCHEMBL22787565 0.74 NAE1 (0.39) AURKANAE1UBA3SAE1UBA2
SCHEMBL24286183 0.72 NAE1 (0.75) AURKARPS6KB1NAE1UBA3
SCHEMBL22787573 0.71 NAE1 (0.52) AURKARPS6KB1NAE1UBA3SAE1
SCHEMBL3461174 0.69 AURKA (0.64) AURKARPS6KB1NAE1UBA3P2RX7
SCHEMBL3461284 0.69 AURKA (0.64) AURKARPS6KB1NAE1UBA3P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249109-A1 TRIAZOLOPYRIMIDINE COMPOUND AND SALT, COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2020-12-17 WO disclosed