SCHEMBL22790109

SCHEMBL22790109

COC(=O)c1cn(C)c2cc(N3CCNCC3)c(F)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 5/20 0.51
LMNA P02545 5/20 0.51
HPGD P15428 4/20 0.51
HSD17B10 Q99714 3/20 0.51
BRD4 O60885 1/20 0.51
TSHR P16473 1/20 0.51
HTT P42858 1/20 0.51
CYP2J2 P51589 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CYP1A2 P05177 1/20 0.48
TOP2A P11388 1/20 0.48
CYP2C9 P11712 1/20 0.48
TOP2B Q02880 1/20 0.48
NR4A2 P43354 7/20 0.44
BRPF1 P55201 1/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22790110 0.81 ALDH1A1 (0.43) KDM4EALDH1A1LMNAHSD17B10HTT
SCHEMBL11392814 0.81 ALDH1A1 (0.74) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL30605634 0.81 ALDH1A1 (0.74) KDM4EALDH1A1LMNAHPGDHSD17B10
Hydrochloric Acid SCHEMBL11026221 0.81 ALDH1A1 (0.73) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL20521397 0.80 KDM4E (0.45) KDM4EALDH1A1LMNAHPGDHSD17B10
Hydrochloric Acid SCHEMBL21832889 0.79 KDM4E (0.47) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22790093 0.79 NR4A2 (0.52) KDM4EALDH1A1LMNAHPGDBRD4
SCHEMBL9634547 0.78 KDM4E (0.79) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL8983611 0.78 KDM4E (0.78) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22790287 0.77 KMT2A (0.42) KDM4ELMNABRD4NR4A2BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249064-A1 COMPOUNDS FOR MODULATING FXR NANJING RUIJIE PHARMA CO., LTD. (CN) 2020-12-17 WO disclosed