SCHEMBL22790239

SCHEMBL22790239

COC(=O)c1cn(S(C(C)C)(C(C)C)C(C)C)c2cc(N3CCNCC3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MMP12 P39900 1/20 0.40
HTR6 P50406 7/20 0.40
KHK P50053 2/20 0.38
SIRT6 Q8N6T7 1/20 0.36
ADRB1 P08588 4/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
NR4A2 P43354 1/20 0.36
MAP2 P11137 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22790093 0.82 NR4A2 (0.52) MEN1KMT2AKDM4EKHKSIRT6
SCHEMBL22790352 0.78 NR4A2 (0.48) MEN1KMT2AKDM4EHTR6KHK
SCHEMBL22790247 0.77 KMT2A (0.44) MEN1KMT2AKDM4ENR4A2
SCHEMBL12306058 0.71 MYC (0.57) MEN1KMT2AKDM4ESIRT6ADRB1
SCHEMBL15547292 0.71 ADRB1 (0.58) MEN1KMT2AKDM4EHTR6SIRT6
SCHEMBL7653332 0.71 ADRB1 (0.58) MEN1KMT2AKDM4EHTR6SIRT6
SCHEMBL1958199 0.70 KDM4E (0.47) MEN1KMT2AKDM4EHTR6SIRT6
SCHEMBL19579582 0.70 ACVR1 (0.51) MEN1KMT2AKDM4ESIRT6ADRB1
SCHEMBL7652198 0.70 ACVR1 (0.47) MEN1KMT2AKDM4ESIRT6ADRB1
SCHEMBL25727525 0.70 KDM4E (0.47) MEN1KMT2AKDM4EHTR6SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249064-A1 COMPOUNDS FOR MODULATING FXR NANJING RUIJIE PHARMA CO., LTD. (CN) 2020-12-17 WO disclosed