SCHEMBL22790352

SCHEMBL22790352

COC(=O)c1cn(C)c2cc(N3CCCNCC3)ccc12

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 8/20 0.48
KHK P50053 4/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
RECQL P46063 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
SIRT6 Q8N6T7 1/20 0.40
BRD4 O60885 1/20 0.39
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22790093 0.95 NR4A2 (0.52) NR4A2KHKMEN1KMT2AKDM4E
SCHEMBL22790131 0.83 SIRT6 (0.56) NR4A2KHKMEN1KMT2AKDM4E
SCHEMBL22790260 0.83 NR4A2 (0.46) NR4A2MEN1KMT2AKDM4ELMNA
SCHEMBL22790174 0.81 NR4A2 (0.47) NR4A2KHKMEN1KMT2AKDM4E
SCHEMBL1096244 0.81 NR4A2 (0.51) NR4A2MEN1KMT2AKDM4ELMNA
SCHEMBL22790129 0.79 NR4A2 (0.49) NR4A2MEN1KMT2AKDM4ELMNA
SCHEMBL22790088 0.78 NR4A2 (0.46) NR4A2MEN1KMT2AKDM4ELMNA
SCHEMBL22789951 0.78 NR4A2 (0.46) NR4A2MEN1KMT2AKDM4ELMNA
SCHEMBL22790239 0.78 MEN1 (0.43) NR4A2KHKMEN1KMT2AKDM4E
SCHEMBL22790343 0.77 KHK (0.46) KHKHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249064-A1 COMPOUNDS FOR MODULATING FXR NANJING RUIJIE PHARMA CO., LTD. (CN) 2020-12-17 WO disclosed