SCHEMBL22790243

SCHEMBL22790243

COC(=O)c1cn([Si](C(C)C)(C(C)C)C(C)C)c2cc(Br)ccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRPS1 P60891 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
NR4A2 P43354 5/20 0.42
KMT2A Q03164 3/20 0.40
MEN1 O00255 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
ELANE P08246 1/20 0.39
CHEK1 O14757 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
THRB P10828 1/20 0.38
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565888 0.81 NR4A2 (0.60) L3MBTL1NR4A2KMT2AMEN1TSHR
SCHEMBL498716 0.80 PRPS1 (0.45) PRPS1L3MBTL1NR4A2KMT2AMEN1
SCHEMBL22790237 0.80 NR4A2 (0.41) L3MBTL1NR4A2KMT2AMEN1ELANE
SCHEMBL497718 0.78 NR4A2 (0.63) PRPS1L3MBTL1NR4A2KMT2AMEN1
SCHEMBL22790247 0.77 KMT2A (0.44) PRPS1L3MBTL1NR4A2KMT2AMEN1
SCHEMBL12127680 0.77 L3MBTL1 (0.37) L3MBTL1NR4A2KMT2AMEN1ALDH1A1
SCHEMBL15025087 0.76 PDGFRA (0.35) CHEK1HTTLMNASMN1; SMN2
SCHEMBL21549969 0.75 NR4A2 (0.66) PRPS1L3MBTL1NR4A2KMT2AMEN1
SCHEMBL35211208 0.75 NR4A2 (0.66) PRPS1L3MBTL1NR4A2KMT2AMEN1
SCHEMBL15024961 0.74 PDGFRA (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249064-A1 COMPOUNDS FOR MODULATING FXR NANJING RUIJIE PHARMA CO., LTD. (CN) 2020-12-17 WO disclosed