SCHEMBL22803045

SCHEMBL22803045

N#CCC(=O)NCc1ccc(Cl)cc1F

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 3/20 0.53
ERCC4 Q92889 3/20 0.53
MCL1 Q07820 1/20 0.48
F2 P00734 1/20 0.44
P2RX7 Q99572 6/20 0.44
ALDH1A1 P00352 1/20 0.43
CNR1 P21554 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
AKR1B1 P15121 3/20 0.41
MMP2 P08253 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2266096 0.85 P2RX7 (0.50) ERCC1ERCC4MCL1P2RX7NPC1
SCHEMBL2265823 0.85 ALDH1A1 (0.58) ERCC1ERCC4MCL1P2RX7ALDH1A1
SCHEMBL2266083 0.83 P2RX7 (0.54) ERCC1ERCC4MCL1F2P2RX7
SCHEMBL23565573 0.82 ERCC1 (0.58) ERCC1ERCC4P2RX7ALDH1A1CNR1
SCHEMBL2263310 0.81 MCL1 (0.51) MCL1P2RX7
SCHEMBL7934896 0.81 ERCC1 (0.57) ERCC1ERCC4P2RX7ALDH1A1CNR1
SCHEMBL2391525 0.81 MCL1 (0.49) ERCC1ERCC4MCL1P2RX7
SCHEMBL2264466 0.80 MCL1 (0.50) ERCC1ERCC4MCL1P2RX7ALDH1A1
SCHEMBL2265012 0.79 MCL1 (0.50) ERCC1ERCC4MCL1P2RX7ALDH1A1
SCHEMBL2266698 0.79 MCL1 (0.61) MCL1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020249821-A1 NOVEL ARGINASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-12-17 WO disclosed