SCHEMBL22809486

SCHEMBL22809486

CC(=O)Nc1cc(C=O)cc(C)n1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
ADORA3 P0DMS8 8/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
ADORA1 P30542 2/20 0.40
ADORA2A P29274 2/20 0.40
LCK P06239 1/20 0.40
ADORA2B P29275 1/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809460 0.82 ADORA3 (0.46) ADORA3ADORA1ADORA2AADORA2BALDH1A1
SCHEMBL18266541 0.82 ADORA3 (0.43) ADORA3ADORA1ADORA2ALCKALDH1A1
SCHEMBL18266627 0.81 HPGD (0.46) ADORA3ADORA1ADORA2AALDH1A1
SCHEMBL50044 0.78 LCK (0.60) PIK3CGL3MBTL1ADORA3CYP1A2LCK
SCHEMBL22809639 0.77 ADORA3 (0.48) ADORA3ADORA1ADORA2AALDH1A1SMN1; SMN2
SCHEMBL23998421 0.75 PIK3CG (0.47) PIK3CGL3MBTL1ADORA3CYP1A2CYP2C9
SCHEMBL16913955 0.75 ADORA3 (0.50) PIK3CGL3MBTL1ADORA3CYP1A2CYP2C9
SCHEMBL29383895 0.75 PIK3CG (0.47) PIK3CGL3MBTL1ADORA3CYP1A2CYP2C9
SCHEMBL13600103 0.75 SRC (0.33) ALDH1A1SMN1; SMN2
SCHEMBL378339 0.74 SRC (0.42) CYP1A2CYP2C19APOBEC3GALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed