SCHEMBL22809583

SCHEMBL22809583

CC(C)(F)c1ccc2nc(OCCN)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.41
SCN9A Q15858 12/20 0.38
HSF1 Q00613 1/20 0.37
SCN7A Q01118 4/20 0.36
KCNH2 Q12809 4/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE7A Q13946 1/20 0.34
SCN5A Q14524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809472 0.89 BACE1 (0.54) BACE1SCN9ASCN7AKCNH2SCN10A
Hydrochloric Acid SCHEMBL20595231 0.87 BACE1 (0.53) BACE1SCN9ASCN7AKCNH2SCN10A
SCHEMBL22809561 0.86 BACE1 (0.41) BACE1SCN9AHSF1SCN7AKCNH2
SCHEMBL22809481 0.74 BACE1 (0.47) BACE1SCN9ASCN7AKCNH2SCN10A
SCHEMBL28350726 0.74 BACE1 (0.47) BACE1SCN9ASCN7AKCNH2SCN10A
SCHEMBL3338851 0.70 TLR8 (0.44) SCN7AKCNH2SCN10A
SCHEMBL28354796 0.69 SCN9A (0.48) SCN9ASCN7AKCNH2SCN10ASCN5A
SCHEMBL19798863 0.66 BACE1 (0.39) BACE1KCNH2SCN10AMEN1KMT2A
SCHEMBL2001524 0.66 HPGD (0.48) SCN9ASMN1; SMN2MAPTKMT2A
SCHEMBL28563865 0.66 ALDH1A1 (0.55) SMN1; SMN2MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed